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Publications

Année 2013 :

1. Omar Aouled, N. O. ; Lebal, N. ; Hallil, H. ; Delépée, R. ; Agrofoglio, L. A. ; Rebière, D. ; Dejous, C.
   Study of gaseous compounds adsorption with a love wave sensor based on Molecularly Imprinted Polymeric thin film
   Sensors & transducers 2013, 149, 37-42.
   
   
2. Sari, O. ; Roy, V. ; Agrofoglio, L. A.
   Nucleosides modified at the base moiety
   Chemical Synthesis of Nucleoside Analogues, P Merino (Ed.); Wiley-VCH GmbH & Co. KgaA (ISBN: 978-1-1180-0751-8), Weinheim 2013, 49-102.
   
   

Année 2012 :

1. Fresneau, N. ; Hiebel, M.-A. ; Agrofoglio, L. A. ; Berteina-Raboin, S.
   One-pot Sonogashira-cyclization protocol to obtain substituted furopyrimidine nucleosides in aqueous conditions
   Tetrahedron Lett. 2012, 53, 1760-1763.
   
   
2. Fresneau, N. ; Hiebel, M.-A. ; Agrofoglio, L. A. ; Berteina-Raboin, S.
   Efficient synthesis of unprotected C-5-aryl/heteroaryl-2'-deoxyuridine via a Suzuki-Miyaura reaction in aqueous media
   Molecules 2012, 17, 4409-14417.
   
   
3. Henry, N. ; Delépée, R. ; Seigneuret, J. M. ; Agrofoglio, L. A.
   Synthesisofwater-compatibleimprintedpolymersof in situ produced fructosazine and 2,5-deoxyfructosazine
   Talanta 2012, 99, 816–823.
   
   
4. Pradère, U. ; Roy, V. ; Montagu, A. ; Sari, O. ; Balzarini, J. ; Snoeck, R. ; Andrei, G. ; Agrofoglio, L. A.
   Synthesis and antiviral evaluation of bis(POM) prodrugs of (E)-[4'-phosphono-but-2'-en-1'-yl]purine nucleosides
   Eur. J. Med. Chem. 2012, 57, 126-133.
   
   
5. Sari, O. ; Roy, V. ; Balzarini, J. ; Snoeck, R. ; Andrei, G. ; Agrofoglio, L. A.
   Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-20-deoxyuridines
   Eur. J. Med. Chem. 2012, 53, 220-228.
   
   

Année 2011 :

1. Montagu, A. ; Roy, V. ; Balzarini, J. ; Snoeck, R. ; Andrei, G. ; Agrofoglio, L. A.
   Synthesis and antiviral evaluation of a series of C5-(1-substituted-1,2,3-triazol-4-yl or 5-yl)-2’-deoxyuridines
   Eur. J. Med. Chem. 2011, 46, 778-786.
   
   
2. Montagu, A. ; Pradère, U. ; Roy, V. ; Nolan, S. P. ; Agrofoglio, L. A.
   Expeditious convergent procedure for the preparation of bis(POC) prodrugs of new (E)-4-phosphono-but-2-en-1-yl nucleosides
   Tetrahedron 2011, 67, 5319-5328.
   
   
3. Pradère, U. ; Clavier, H. ; Roy, V. ; Nolan, S. P. ; Agrofoglio, L. A.
   The shortest strategy for generating phosphonate prodrugs by olefin cross-metathesis – application to acyclonucleoside phosphonates
   Eur. J. Org. Chem. 2011, 7324-7330.
   
   
4. Roy, V. ; Li, Y. ; Obikhod, A. ; Zhang, H.-W. ; Coats, S. J. ; Herman, B. D. ; Sluis-Cremer, N. ; Agrofoglio, L. A. ; Schinazi, R.F.
   Synthesis and anti-HIV evaluation of 3’-triazolo nucleosides
   Nucleosides Nucleotides Nucleic Acids 2011, 30, 264-270.
   
   
5. Roy, V. ; Pradère, U. ; Montagu, A. ; Nolan, S. P. ; Agrofoglio, L. A.
   Phosphonate synthons bearing a biolabile group for olefin cross metathesis: synthesis of acyclonucleoside phosphonate analogs
   Collection Symposium Series (2011) Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, Prague 2011, 12, 213-217.
   
   
6. Salwiński, A. ; Roy, V. ; Agrofoglio, L. A. ; Delépée, R.
   In situ one-step method for synthesis of “click”-functionalized monolithic stationary phase for capillary electrochromatography
   Macromolecular Chemistry and Physics 2011, 212, 2700-2707.
   
   
7. Topalis, D. ; Pradère, U. ; Roy, V. ; Caillat, C. ; Azzouzi, A. ; Broggi, J. ; Snoeck, R. ; Andrei, G. ; Lin, J. ; Eriksson, S. ; Alexandre, J.A.C. ; El Amri, C. ; Deville-Bonne, D. ; Meyer, P. ; Balzarini, J. ; Agrofoglio, L. A.
   Novel antiviral C5-substituted pyrimidine acyclic nucleoside phosphonates selected as human YMP kinase substrates
   J. Med. Chem. 2011, 54, 222-232.
   
   

Année 2010 :

1. Deville-Bonne, D. ; El Amri, C. ; Meyer, P. ; Chen Y. ; Agrofoglio, L. A. ; Janin J.
   Human and viral nucleoside/nucleotide kinases involved in antiviral drug activation: Structural and catalytic properties
   Antiviral Research 2010, 86, 101-120.
   
   
2. Lin, J. ; Roy, V. ; Wang, L. ; You, L. ; Agrofoglio, L. A. ; Deville-Bonne, D. ; McBrayer, T. R. ; Coats, S. J. ; Schinazi, R.F. ; Eriksson, S.
   3´-(1,2,3-triazol-1-yl)-3’-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure-activity investigations
   Bioorg. Med. Chem. 2010, 18, 3261-3269.
   
   
3. Mieczkowski, A. ; Roy, V. ; Agrofoglio, L. A.
   Preparation of cyclonucleosides
   Chemical Reviews 2010, 110, 1828-1856.
   
   
4. Mieczkowski, A. ; Agrofoglio, L. A.
   Potential and perspectives of cyclonucleosides
   Current Medicinal Chemistry 2010, 17, 1527-1549.
   
   
5. Pradère, U. ; Kumamoto, H. ; Roy, V. ; Agrofoglio, L. A.
   Preparation of carbocyclic C-nucleosides from a-chlorooxime precursor
   Eur. J. Org. Chem. 2010, 2010, 749-754.
   
   
6. Roy, V. ; Pradère, U. ; Agrofoglio, L. A.
   Microwave-assisted syntheses of nucleosides and their precursors
   Future Med. Chem. 2010, 2, 177-192.
   
   

Année 2009 :

1. Auvynet, C. ; Topalis, D. ; Caillat, C. ; Munier-Lehmann, H. ; Seclaman, E. ; Balzarini, J. ; Agrofoglio, L. A. ; Kaminski, P. A. ; Meyer, P. ; Deville-Bonne, D. ; El Amri, C.
   Phosphorylation of dGMP analogs by vaccinia virus TMP kinase and human GMP kinase
   Biochemical and Biophysical Research Communications 2009, 388, 6-11.
   
   
2. Breton, F. ; Delépée, R. ; Agrofoglio, L. A.
   Molecular imprinting of AMP by an ionic-noncovalent dual approach
   Journal of Separation Science 2009, 32, 3285-3291.
   
   
3. Broggi, J. ; Joubert, N. ; Díez-González , S. ; Berteina-Raboin, S. ; Zevaco, T. ; Nolan, S. P. ; Agrofoglio, L. A.
   Synthesis of (±)-1,2,3-triazolo-3'-deoxy-4'-hydroxymethyl carbanucleosides via ‘click’ cycloaddition
   Tetrahedron 2009, 65, 1162-1170.
   
   
4. Broggi, J. ; Kumamoto, H. ; Berteina-Raboin, S. ; Nolan, S. P. ; Agrofoglio, L. A.
   Click azide-alkyne cycloaddition for the synthesis of D-(-)-1,4-disubstituted triazolo-carbanucleosides
   Eur. J. Org. Chem. 2009, 2009, 1880-1888.
   
   
5. Mieczkowski, A. ; Peltier, P. ; Zevaco, T. ; Agrofoglio, L. A.
   Preparation of C5-substituted O⁶,5'-cyclouridine
   Tetrahedron 2009, 65, 4053-4059.
   
   
6. Mieczkowski, A. ; Blu, J. ; Roy, V. ; Agrofoglio, L. A.
   Preparation of C-5-substituted 6,5'-O-anhydrouridine by Sn–Pd transmetallation-coupling process and their use
   Tetrahedron 2009, 65, 9791–9796.
   
   

Année 2008 :

1. Agrofoglio, L. A. ; Mieczkowski, A.
   Synthesis and biological activity of selected carbocyclic nucleosides
   Modifed Nucleosides in Biochemistry, Biotechnology and Medecine ; P Herdewijn (Ed.); Wiley-VCH GmbH & Co. KgaA, Weinheim 2008, .
   
   
2. Breton, F. ; Delépée, R. ; Jégourel, D. ; Deville-Bonne, D. ; Agrofoglio, L. A.
   Selective adenosine-5'-monophosphate uptake by water-compatible molecularly imprinted polymer
   Anal. Chim. Acta 2008, 616, 222-229.
   
   
3. Broggi, J. ; Díez-González , S. ; Petersen, J. L. ; Berteina-Raboin, S. ; Nolan, S. ; Agrofoglio, L. A.
   Study of copper(I) catalysts for the synthesis of carbanucleosides via azide-alkyne 1,3-dipolar cycloaddition
   Synthesis 2008, 141-148.
   
   
4. Caillat, C. ; Topalis, D. ; Agrofoglio, L. A. ; Pochet, S. ; Balzarini, J. ; Deville-Bonne, D. ; Meyer, P.
   Crystal structure of poxvirus thymidylate kinase shows an unexpected dimerization with implication for antiviral therapy
   Proceedings of the National Academy of Sciences 2008, 105, 16900-16905.
   
   
5. Delépée, R. ; Got, L. ; Causse, X. ; Agrofoglio, L. A. ; Si Ahmed S. N.
   Simultaneous determination of tenofovir, adefovir, lamivudine, entecavir in plasma
   Journal of Hepatology - Abstracts of the 43rd Annual Meeting of the European Association for the Study of the Liver 2008, 48, S215-S216.
   
   
6. Jégourel, D. ; Delépée, R. ; Breton, F. ; Rolland, A. ; Vidal, R. ; Agrofoglio, L. A.
   Molecularly imprinted polymer of 5-methyluridine for solid-phase extraction of pyrimidine nucleoside cancer markers in urine
   Bioorg. Med. Chem. 2008, 16, 8932-8939.
   
   
7. Joubert, N. ; Amblard, F. ; Rapp, K. L. ; Schinazi, R.F. ; Agrofoglio, L. A.
   Synthesis and anti-HIV activity of 5-haloethynyl- and 5-(1,2-Dihalo)vinyl Analogues of AZT and FLT
   Tetrahedron 2008, 64, 4444-4452.
   
   
8. Kumamoto, H. ; Topalis, D. ; Broggi, J. ; Pradère, U. ; Roy, V. ; Berteina-Raboin, S. ; Nolan, S. P. ; Deville-Bonne, D. ; Snoeck, R. ; Garin, D. ; Crance, J. M. ; Agrofoglio, L. A.
   Preparation of acyclo nucleoside phosphonate analogues based-on cross-metathesis
   Tetrahedron 2008, 64, 3517-3526.
   
   
9. Pradère, U. ; Roy, V. ; McBrayer, T. R. ; Schinazi, R.F. ; Agrofoglio, L. A.
   Preparation of ribavirin analogues by copper- and ruthenium-catalyzed azide-alkyne 1,3-dipolar cycloaddition
   Tetrahedron 2008, 64, 9044-9051.
   
   
10. Pruvost, A. ; Théodoro, F. ; Levi, M. ; Agrofoglio, L. A. ; Negredo, E. ; Benech, H.
    Specificity enhancement with LC-positive ionization ESI-MS/MS for the measurement of nucleotides : Application to the quantitative determination of carbovir triphosphate, lamivudine triphosphate and tenofovir diphosphate in human peripheral blood mononuclear cells.
    Journal of Mass Spectrometry 2008, 43, 224-233.
    
    
11. Roy, V. ; Mieczkowski, A. ; Topalis, D. ; Berteina-Raboin, S. ; Deville-Bonne, D. ; Nolan, S. P. ; Agrofoglio, L. A.
    Microwave-assisted silylation-amination of uracil acyclonucleosides to 4-alkylamino-2(1H)-pyrimidinone analogues
    Synthesis 2008, 2127-2133.
    
    
12. Topalis, D. ; Broggi, J. ; Alexandre, J.A.C. ; Pradère, U. ; Roy, V. ; Berteina-Raboin, S. ; Agrofoglio, L. A. ; Deville-Bonne, D.
    Evaluation of C-5 substituted uracil acyclic phosphonates as substrates or inhibitors for DTMP and UMP–CMP kinases and potential antipox derivatives
    Antiviral Research 2008, 78, A65.
    
    

Année 2007 :

1. Agrofoglio, L. A. ; Amblard, F. ; Broggi, J. ; Garnier, E.
   Recent insights into the synthesis of "non-classical" O- and N-heterocyclic bases of nucleosides
   in Modern Approaches to the Synthesis of O- and N-Heterocyles Eds.: Kaufman TS and Larghi EL, Research Signpost, Trivandrum, India 2007, 2, 195-246.
   
   
2. Agrofoglio, L. A. ; Bezy, V. ; Chaimbault, P. ; Delépée, R. ; Rhourri, B. ; Morin, Ph.
   Mass spectrometry based methods for analysis of nucleosides as antiviral drugs and potential tumor biomarkers
   Nucleosides Nucleotides Nucleic Acids 2007, 26, 1523-1527.
   
   
3. Broggi, J. ; Joubert, N. ; Aucagne, V. ; Zevaco, T. ; Berteina-Raboin, S. ; Nolan, S. P. ; Agrofoglio, L. A.
   Study of different copper (I) catalysts for the "click chemistry" approach to carbanucleosides
   Nucleosides Nucleotides Nucleic Acids 2007, 26, 779-783.
   
   
4. Broggi, J. ; Joubert, N. ; Aucagne, V. ; Berteina-Raboin, S. ; Diez-Gonzales, S. ; Nolan, S. ; Topalis, D. ; Deville-Bonne, D. ; Balzarini, J. ; Neyts, J. ; Andrei, G. ; Snoeck, R. ; Agrofoglio, L. A.
   Alkyne-azide click chemistry mediated carbanucleosides synthesis
   Nucleosides Nucleotides Nucleic Acids 2007, 26, 1391-1394.
   
   
5. El Kazzouli, S. ; Berteina-Raboin, S. ; Agrofoglio, L. A.
   Supported synthesis and functionnalization of 2"-deoxyuridine by suzuki-miyaura cross-coupling
   Nucleosides Nucleotides Nucleic Acids 2007, 26, 1395-1398.
   
   
6. Roy, V. ; Kumamoto, H. ; Berteina-Raboin, S. ; Nolan, S. P. ; Topalis, D. ; Deville-Bonne, D. ; Balzarini, J. ; Neyts, J. ; Andrei, G. ; Snoeck, R. ; Agrofoglio, L. A.
   Cross-metathesis mediated synthesis of new acyclic nucleoside phosphonates
   Nucleosides Nucleotides Nucleic Acids 2007, 26, 1399-1402.
   
   
7. Topalis, D. ; Kumamoto, H. ; Amaya Velasco, M.-F. ; Dugué, L. ; Haouz, A. ; Alexandre, J.A.C. ; Gallois-Montbrun S. ; Alzari P.M. ; Pochet, S. ; Agrofoglio, L. A. ; Deville-Bonne, D.
   Nucleotide binding to human UMP-CMP kinase using fluorescent derivatives: a screenin approach based on afinity for UMP-CMP binding site
   FEBS Journal 2007, 274, 3704-3714.
   
   
8. Topalis, D. ; Kumamoto, H. ; Alexandre, J. A. ; Dugué, L. ; Pochet, S. ; Berteina-Raboin, S. ; Agrofoglio, L. A. ; Deville-Bonne, D.
   Looking for new pyrimidine acyclic nucleotide analogues designed for phosphorylation by human ump-cmp kinase
   Nucleosides Nucleotides Nucleic Acids 2007, 26, 1369-1373.
   
   

Année 2006 :

1. Agrofoglio, L. A. ; Joubert, N. ; Escuret, V. ; Durantel, D. ; Zoulim, F.
   The use of the HCV replicon system for the evaluation of new nucleoside analogs
   Framing the Knowledge of Therapeutics for Viral Hepatitis, Ed. RF Schinazi and ER Schiff [v-vii], IHL Press 2006, 183-196.
   
   
2. Agrofoglio, L. A.
   An overview of diazine nucleoside analogues
   Current Organic Chemistry 2006, 10, 333-362.
   
   
3. Agrofoglio, L. A. ; Kumamoto, H. ; Roy, V.
   Cross-metathesis in the synthesis of bioactive phosphonates
   Chemistry Today 2006, 24, 16-18.
   
   
4. Bezy, V. ; Chaimbault, P. ; Morin, Ph. ; Unger, S. E. ; Bernard, M. C. ; Agrofoglio, L. A.
   Analysis and validation of the phosphorylated metabolites of two anti-HIV nucleotides by pressure-assisted CE/ESI-MS/MS in cell extracts. Sensitivity enhancement by the use of perfluorinated acids and alcohols as coaxial sheath liquid makue-up constituents
   Electrophoresis 2006, 27, 2464-2476.
   
   

Année 2005 :

1. Agrofoglio, L. A. ; Nolan, S. P.
   Olefin metathesis route to antiviral nucleosides
   Curr. Top. Med. Chem. 2005, 5, 1541-1558.
   
   
2. Amblard, F. ; Nolan, S. P. ; Schinazi, R.F. ; Agrofoglio, L. A.
   Efficient synthesis of various acycloalkenyl derivatives of pyrimidine using cross-metathesis and Pd(0) methodologies
   Tetrahedron 2005, 61, 537-544.
   
   
3. Amblard, F. ; Aucagne, V. ; Guenot, P. ; Schinazi, R.F. ; Agrofoglio, L. A.
   Synthesis and antiviral activity of novel acyclic nucleosides in the 5-alkynyl and 6-alkylfuro[2,3-d]pyrimidine series
   Bioorg. Med. Chem. 2005, 13, 1239-1248.
   
   
4. Amblard, F. ; Nolan, S. P. ; Agrofoglio, L. A.
   Metathesis strategy in nucleoside chemistry
   Tetrahedron 2005, 61, 7067-7080.
   
   
5. Bezy, V. ; Morin, Ph. ; Couerbe Ph. ; Leleu G. ; Agrofoglio, L. A.
   Simultaneous analysis of several antiretroviral nucleosides in rat-plasma by high-performance liquid chromatography with UV using acetic acid/hydroxylamine buffer . Test of this new volatile medium-pH for HPLC-ESI-MS/MS
   Journal of Chromatography B 2005, 821, 132-143.
   
   
6. Escuret, V. ; Aucagne, V. ; Joubert, N. ; Durantel, D. ; Rapp, K. L. ; Schinazi, R.F. ; Zoulim, F. ; Agrofoglio, L. A.
   Synthesis of 5-haloethynyl- and 5-(1,2-dihalo)vinyluracil nucleosides : Antiviral activity and cellular toxicity
   Bioorg. Med. Chem. 2005, 13, 6015-6024.
   
   
7. Joubert, N. ; Schinazi, R.F. ; Agrofoglio, L. A.
   Efficient Pd(0)-catalyzed synthesis of 1,2,3-triazolo-3'-deoxycarbanucleosides and their analogues
   Tetrahedron 2005, 61, 11744-11750.
   
   

Année 2004 :

1. Agrofoglio, L. A. ; Amblard, F. ; Nolan, S. P. ; Charamon, S. ; Gillaizeau, I. ; Zevaco, T. A. ; Guenot, P.
   Synthesis of L-cyclopentenyl nucleosides using ring-closing metathesis and palladium-mediated allylic alkylation methodologies
   Tetrahedron 2004, 60, 8397-8404.
   
   
2. Aucagne, V. ; Berteina-Raboin, S. ; Guenot, P. ; Agrofoglio, L. A.
   Palladium-catalyzed parallel solid-phase synthesis of nucleosides
   Journal of Combinatorial Chemistry 2004, 6, 717-723.
   
   
3. Aucagne, V. ; Amblard, F. ; Agrofoglio, L. A.
   Highly efficient AgNO₃-catalyzed preparation of substituted furanopyrimidine nucleosides
   Synlett 2004, 2406-2410.
   
   

Année 2003 :

1. Agrofoglio, L. A. ; Gillaizeau, I. ; Saito, Y.
   Palladium-assisted routes to nucleosides
   Chemical Reviews 2003, 103, 1875-1916.
   
   
2. Amblard, F. ; Nolan, S. P. ; Gillaizeau, I. ; Agrofoglio, L. A.
   A new route to acyclic nucleosides via palladium-mediated allylic alkylation and cross-metathesis
   Tetrahedron Lett. 2003, 44, 9177-9180.
   
   
3. Gillaizeau, I. ; Lagoja, I. M. ; Nolan, S. P. ; Aucagne, V. ; Rozenski, J. ; Herdewijn, P. ; Agrofoglio, L. A.
   Straightforward synthesis of labeled and unlabeled pyrimidine d4Ns via 2',3'-diyne seco analogues through olefin metathesis reactions
   Eur. J. Org. Chem. 2003, 4, 666-671.
   
   
4. Mesplet, N. ; Saito, Y. ; Morin, Ph. ; Agrofoglio, L. A.
   Liquid chromatographic separation of phosphoramidates diastereomers on a polysaccharide-type chiral stationary phase
   J. Chromatogr. A 2003, 983, 115-124.
   
   
5. Mesplet, N. ; Saito, Y. ; Morin, Ph. ; Agrofoglio, L. A.
   HPLC and mass spectrometry analysis of the enzymatic hydrolysis of anti-HIV pronucleotide diastereomers
   Bioorganic Chemistry 2003, 31, 237-247.
   
   
6. Saito, Y. ; Escuret, V. ; Durantel, D. ; Zoulim, F. ; Schinazi, R.F. ; Agrofoglio, L. A.
   Synthesis of 1,2,3-triazolo-carbanucleoside analogues of ribavirin targeting an HCV in replicon
   Bioorg. Med. Chem. 2003, 11, 3633-3639.
   
   

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